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Academic Journal

A Novel and Selective Dopamine Transporter Inhibitor, (S) -MK-26, Promotes Hippocampal Synaptic Plasticity and Restores Effort-Related Motivational Dysfunctions.

  • Authors : Kouhnavardi S; Programme for Proteomics, Paracelsus Medical University, 5020 Salzburg, Austria.; Department of Pharmaceutical Chemistry, Faculty of Life Sciences, University of Vienna, 1090 Vienna, Austria.

Subjects: Dopamine* ; Dopamine Plasma Membrane Transport Proteins*/Dopamine Plasma Membrane Transport Proteins*/Dopamine Plasma Membrane Transport Proteins*/antagonists & inhibitors ; Dopamine Plasma Membrane Transport Proteins*/Dopamine Plasma Membrane Transport Proteins*/Dopamine Plasma Membrane Transport Proteins*/metabolism

  • Source: Biomolecules [Biomolecules] 2022 Jun 24; Vol. 12 (7). Date of Electronic Publication: 2022 Jun 24.Publisher: MDPI Country of Publication: Switzerland NLM ID: 101596414 Publication Model: Electronic Cited Medium: Internet ISSN: 2218-273X

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Periodical

Reinstatement of synaptic plasticity in the aging brain through specific dopamine transporter inhibition.

  • Authors : Lubec J; Programme for Proteomics, Paracelsus Medical University, Salzburg, Austria.; Kalaba P

Subjects: Dopamine Plasma Membrane Transport Proteins* ; Neuronal Plasticity*/Neuronal Plasticity*/Neuronal Plasticity*/physiology; Aging

  • Source: Molecular psychiatry [Mol Psychiatry] 2021 Dec; Vol. 26 (12), pp. 7076-7090.Publisher: Nature Publishing Group Specialist Journals Country of Publication: England NLM ID: 9607835 Publication Model: Print Cited Medium: Internet

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Academic Journal

Structure-Activity Relationships of Novel Thiazole-Based Modafinil Analogues Acting at Monoamine Transporters.

  • Authors : Kalaba P; Department of Pharmaceutical Chemistry, Faculty of Life Sciences , University of Vienna , Althanstraße 14 , 1090 Vienna , Austria.; Ilić M

Subjects: Dopamine Plasma Membrane Transport Proteins/Dopamine Plasma Membrane Transport Proteins/Dopamine Plasma Membrane Transport Proteins/*antagonists & inhibitors ; Dopamine Uptake Inhibitors/Dopamine Uptake Inhibitors/Dopamine Uptake Inhibitors/*pharmacology ; Modafinil/Modafinil/Modafinil/*analogs & derivatives

  • Source: Journal of medicinal chemistry [J Med Chem] 2020 Jan 09; Vol. 63 (1), pp. 391-417. Date of Electronic Publication: 2019 Dec 30.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

Heterocyclic Analogues of Modafinil as Novel, Atypical Dopamine Transporter Inhibitors.

  • Authors : Kalaba P; Department of Pharmaceutical Chemistry, Faculty of Life Sciences, University of Vienna , Althanstraße 14, 1090 Vienna, Austria.; Aher NY

Subjects: Benzhydryl Compounds/Benzhydryl Compounds/Benzhydryl Compounds/*pharmacology ; Dopamine Plasma Membrane Transport Proteins/Dopamine Plasma Membrane Transport Proteins/Dopamine Plasma Membrane Transport Proteins/*antagonists & inhibitors ; Dopamine Uptake Inhibitors/Dopamine Uptake Inhibitors/Dopamine Uptake Inhibitors/*pharmacology

  • Source: Journal of medicinal chemistry [J Med Chem] 2017 Nov 22; Vol. 60 (22), pp. 9330-9348. Date of Electronic Publication: 2017 Nov 09.Publisher: American Chemical Society Country of Publication: United States NLM ID: 9716531 Publication Model: Print-Electronic Cited Medium: Internet

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Academic Journal

A novel heterocyclic compound targeting the dopamine transporter improves performance in the radial arm maze and modulates dopamine receptors D1-D3.

  • Authors : Saroja SR; Department of Pediatrics, Medical University of Vienna, 1090 Vienna, Austria; Department of Cell Biology, Duke University School of Medicine, NC 27710, USA.

Subjects: Benzhydryl Compounds/Benzhydryl Compounds/Benzhydryl Compounds/*administration & dosage ; Benzhydryl Compounds/Benzhydryl Compounds/Benzhydryl Compounds/*pharmacokinetics ; Benzhydryl Compounds/Benzhydryl Compounds/Benzhydryl Compounds/*pharmacology

  • Source: Behavioural brain research [Behav Brain Res] 2016 Oct 01; Vol. 312, pp. 127-37. Date of Electronic Publication: 2016 Jun 08.Publisher: Elsevier/North-Holland Biomedical Press Country of Publication: Netherlands NLM ID: 8004872 Publication Model: Print-Electronic Cited Medium:

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